KISS1R / GPR54 Activation
GPR54 Agonist
Binds KISS1R on GnRH neurons in the hypothalamus. The receptor sits upstream of the reproductive axis rather than within the gonads, which is what makes the peptide useful for studying regulation rather than output.
- Binds KISS1R on hypothalamic GnRH neurons
- Acts upstream of the gonads, not on them
- Ten-residue active fragment of kisspeptin-54






